Acetyl-(D-Arg10 Cys11 D-Phe1, Each

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Acetyl-(D-Arg10,Cys11,D-Phe14,Cys17) 5Mg Highly Potent And Selective ª-Msh-Derived Melanocortin-4 Receptor (Mc-4R) Agonist With Sub-Nanomolar Potency. The Binding Affinities For Human Mc-4R, Mc-1R, Mc-3R And Mc-5R Were 0.55 ª 0.06, 16.78 ª 1.53, 56.79 ª 4.66, And < 500 Nm, Respectively. Daily Subcutaneous Injection Of H-6268 To Diet-Induced Obese Rats Over A Period Of 14 Days Demonstrated An Effect On Reduction Of Fat Mass. (Disulfide Bond) Cas: 819048-44-7 C51H70N18O11S2 Fw: 1175.36. Msh