Calbiochem InSolution 1-Azakenpaullone, A Kenpaullone analog that acts as a potent and ATP-competitive inhibitor of GSK-3andbeta, Each

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A Kenpaullone (Cat. No. 422000) analog that acts as a potent and ATP-competitive inhibitor of GSK-3β (IC50 = 18nM). Displays over 100-fold greater selectivity over Cdk1/cyclin B and Cdk5/p25 (IC50 = 2.0μM and 4.2μM, respectively). The solid form of this compound (Cat. No. 191500) is also available.