ERK5-IN-1, Potent and selective ERK5 inhibitor, Each
$ 3,120.86
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Details
ERK5-IN-1 is a potent and selective ERK5 inhibitor; inhibits EGFR-induced ERK5 autophosphorylation (EC50 = 90 nM) and ERK5 enzymatic activity (IC50 = 162 nM). Exhibits at least 30-fold selectivity for ERK5 over LRRK2 in a cell based assay. Also selective for ERK5 over a panel of other kinases. Orally bioavailable.
Additional Information
| SKU | 10263760 |
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| UOM | Each |
| UNSPSC | 41116105 |
| Manufacturer Part Number | 5393/50 |
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