GSK 5959, Potent and selective BRPF1 inhibitor, Each
$ 434.19
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Details
GSK 5959 is a potent and selective BRPF1 bromodomain inhibitor (IC50 = 80 nM). Exhibits >100-fold selectivity for BRPF1 over a panel of 35 other bromodomains, including BRPF2/3 and BET family bromodomains. Inhibits BRPF1 interaction with histone H3.3. Cell permeable.
Additional Information
SKU | 10509008 |
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UOM | Each |
UNSPSC | 41116105 |
Manufacturer Part Number | 5385/10 |