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GSK 5959, Potent and selective BRPF1 inhibitor, Each

434.19

Details

GSK 5959 is a potent and selective BRPF1 bromodomain inhibitor (IC50 = 80 nM). Exhibits >100-fold selectivity for BRPF1 over a panel of 35 other bromodomains, including BRPF2/3 and BET family bromodomains. Inhibits BRPF1 interaction with histone H3.3. Cell permeable.

Additional Information

SKU 10509008
UOM Each
UNSPSC 41116105
Manufacturer Part Number 5385/10